Definition of ZD4054

An orally available selective antagonist of the endothelin-A (ET-A) receptor with potential antineoplastic activity. ZD4054 binds selectively to the ET-A receptor, thereby inhibiting endothelin-mediated mechanisms that promote tumor cell proliferation. (NCI05)

ZD4054 is from the group

Endothelin Receptor Antagonist

Other Names for ZD4054



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